ChemInform Abstract: Chiral Broensted Acid-Catalyzed Alkylation of C3-Substituted Indoles with o-Hydroxybenzyl Alcohols: Highly Enantioselective Synthesis of Diarylindol-2-ylmethanes and Evaluation on Their Cytotoxicity.
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- 作者：Qiong Wu ; Chun Ma ; Xi-hua Du ; Yan Chen ; Tian-zi Huang ; Xiao-qin Shi ; Shu-jiang Tu and Pei-jun Cai
- 刊名：ChemInform
- 出版年：2016
- 出版时间：July, 2016
- 年：2016
- 卷：47
- 期：33
- 全文大小：27K
- ISSN：1522-2667
文摘
A chiral phosphoric acid catalyzed Friedel—Crafts alkylation of 2-hydroxybenzyl alcohols (I) with 3-methylindols (II) and (IV) is established.