Palladium-Catalyzed Direct and Regioselective C鈭扝 Bond Functionalization/Oxidative Acetoxylation of Indoles

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• 作者：Pui Ying Choy ; Chak Po Lau ; Fuk Yee Kwong
• 刊名：Journal of Organic Chemistry
• 出版年：2011
• 出版时间：January 7, 2011
• 年：2011
• 卷：76
• 期：1
• 页码：80-84
• 全文大小：824K
• 年卷期：v.76,no.1(January 7, 2011)
• ISSN：1520-6904

文摘

The first general examples of palladium-catalyzed direct and selective oxidative C3-acetoxylation of indoles are presented. The mild reaction conditions (70 掳C and with weak base, KOAc) in this indole C鈭扝-acetoxylation are notable.