Synthesis of α-Aminonaphthalenes via Copper-Catalyzed Aminobenzannulation of (o-Alkynyl)arylketones with Amines

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• 作者：Mingliang Zhang ; Wenqing Ruan ; Hui-Jun Zhang ; Weiwei Li ; Ting-Bin Wen
• 刊名：Journal of Organic Chemistry
• 出版年：2016
• 出版时间：February 19, 2016
• 年：2016
• 卷：81
• 期：4
• 页码：1696-1703
• 全文大小：535K
• ISSN：1520-6904

文摘

A copper-catalyzed aminobenzannulation of (o-alkynyl)arylketones with amines has been developed. This method features the use of a cheap copper catalyst, the facile annulation involving various amines, and the good functional group tolerance.