Tumor Targeting with Novel 6-Substituted Pyrrolo [2,3-d] Pyrimidine Antifolates with Heteroatom Bridge Substitutions via Cellular Uptake by Folate Receptor α and the Proton-Coupled Folate Transporter and Inhibition of de Novo Purine Nucleotide Biosynthesis

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• 作者：Lalit K. Golani ; Adrianne Wallace-Povirk ; Siobhan M. Deis ; Jennifer Wong ; Jiyuan Ke ; Xin Gu ; Sudhir Raghavan ; Mike R. Wilson ; Xinxin Li ; Lisa Polin ; Parker W. de Waal ; Kathryn White ; Juiwanna Kushner ; Carrie O’Connor ; Zhanjun Hou ; H. Eric Xu ; Karsten Melcher ; Charles E. Dann III ; Larry H. Matherly ; Aleem Gangjee
• 刊名：Journal of Medicinal Chemistry
• 出版年：2016
• 出版时间：September 8, 2016
• 年：2016
• 卷：59
• 期：17
• 页码：7856-7876
• 全文大小：1011K
• 参考文献：
• ISSN：1520-4804

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