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Wiley电子期刊(5)	NATURE电子期刊(2)	ACS电子期刊(22)
SpringerLink电子期刊(16)	Elsevier电子期刊(114)

在“Elsevier电子期刊”中，命中：114条，耗时：0.0339833 秒

在所有数据库中总计命中：159条

1.Discovery of novel piperidine-substituted indolylarylsulfones as potent HIV NNRTIs via structure-guided scaffold morphing and fragment rearrangement

作者：Xiao Li^a ; Ping Gao^a ; Boshi Huang^a ; Zhongxia Zhou^a ; Zhao Yu^a ; Zheng Yuan^c ; Huiqing Liu^c ; Christophe Pannecouque^b ; Dirk Daelemans^b ; Erik De Clercq^b ; Peng Zhan^a ; ^{zhanpeng1982@sdu.edu.cn} ; Xinyong Liu^a ; ^{xinyongl@sdu.edu.cn}

关键词：HIV ; NNRTIs ; Indolylarylsulfones ; Antiviral activity ; SAR ; Molecular modeling ; Chemical space ; Drug design

刊名：European Journal of Medicinal Chemistry

出版年：2017

2.Design, synthesis and evaluation of novel HIV-1 NNRTIs with dual structural conformations targeting the entrance channel of the NNRTI binding pocket

作者：Qing Meng^a ; Xuwang Chen^a ; Dongwei Kang^a ; Boshi Huang^a ; Wenxin Li^a ; Peng Zhan^a ; Dirk Daelemans^b ; Erik De Clercq^b ; Christophe Pannecouque^b ; ^{Christophe.Pannecouque@rega.kuleuven.be" class="auth_mail" title="E-mail the corresponding author} ; Xinyong Liu^a ; ^{xinyongl@sdu.edu.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：HIV-1 NNRTIs ; DAPY derivatives ; Dual structural conformations ; Entrance channel ; SARs

刊名：European Journal of Medicinal Chemistry

出版年：2016

3.Design, synthesis and anti-HIV evaluation of novel diarylpyridine derivatives targeting the entrance channel of NNRTI binding pocket

作者：Jiapei Yang^a ; Wenmin Chen^a ; Dongwei Kang^a ; Xueyi Lu^a ; Xiao Li^a ; Zhaoqiang Liu^a ; Boshi Huang^a ; Dirk Daelemans^b ; Christophe Pannecouque^b ; Erik De Clercq^b ; Peng Zhan^a ; ^{zhanpeng1982@sdu.edu.cn" class="auth_mail" title="E-mail the corresponding author} ; Xinyong Liu^a ; ^{xinyongl@sdu.edu.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：HIV-1 ; NNRTIs ; DAPY ; Molecular hybridization ; Drug design ; Entrance channel

刊名：European Journal of Medicinal Chemistry

出版年：2016

4.Modification of the length and structure of the linker of N⁶-benzyladenosine modulates its selective antiviral activity against enterovirus 71

作者：Mikhail S. Drenichev^a ; ¹ ; Vladimir E. Oslovsky^a ; ¹ ; Liang Sun^b ; Aloys Tijsma^b ; Nikolay N. Kurochkin^a ; Vitali I. Tararov^a ; Alexander O. Chizhov^c ; Johan Neyts^b ; Christophe Pannecouque^b ; Pieter Leyssen^b ; Sergey N. Mikhailov^a ; ^{smikh@eimb.ru" class="auth_mail" title="E-mail the corresponding author}

关键词：N6-benzyladenosine derivatives ; Synthesis and antiviral activity ; SAR ; Enterovirus 71

刊名：European Journal of Medicinal Chemistry

出版年：2016

5.Arylazolyl(azinyl)thioacetanilides. Part 20: Discovery of novel purinylthioacetanilides derivatives as potent HIV-1 NNRTIs via a structure-based bioisosterism approach

作者：Xueyi Lu^a ; Xiao Li^a ; Jiapei Yang^a ; Boshi Huang^a ; Dongwei Kang^a ; Fabao Zhao^a ; Zhongxia Zhou^a ; Erik De Clercq^b ; Dirk Daelemans^b ; Christophe Pannecouque^b ; ^{Christophe.Pannecouque@rega.kuleuven.be" class="auth_mail" title="E-mail the corresponding author} ; Peng Zhan^a ; ^{zhanpeng1982@sdu.edu.cn" class="auth_mail" title="E-mail the corresponding author} ; Xinyong Liu^a ; ^{xinyongl@sdu.edu.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：HIV-1 ; AIDS ; NNRTIs ; Purinylthioacetanilide ; Anti-HIV activity ; Drug design ; Bioisosterism

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

6.Structural optimization of pyridine-type DAPY derivatives to exploit the tolerant regions of the NNRTI binding pocket

作者：Wenmin Chen^a ; Peng Zhan^a ; Dirk Daelemans^b ; Jiapei Yang^a ; Boshi Huang^a ; Erik De Clercq^b ; Christophe Pannecouque^b ; ^{Christophe.Pannecouque@rega.kuleuven.be" class="auth_mail" title="E-mail the corresponding author} ; Xinyong Liu^a ; ^{xinyongl@sdu.edu.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：Piperidyl ; Morpholinyl ; Pyridine ; Diarylpyrimidines ; NNRTI ; HIV

刊名：European Journal of Medicinal Chemistry

出版年：2016

7.The G-quadruplex-forming aptamer AS1411 potently inhibits HIV-1 attachment to the host cell

作者：Rosalba Perrone^a ; Elena Butovskaya^a ; Sara Lago^a ; Alfredo Garzino-Demo^a ; ^b ; Christophe Pannecouque^c ; Giorgio Palù ; ^a ; Sara N. Richter^a ; ^{sara.richter@unipd.it" class="auth_mail" title="E-mail the corresponding author}

关键词：HIV ; Aptamer ; Antiretroviral drug ; Attachment

刊名：International Journal of Antimicrobial Agents

出版年：2016

8.1,6-Bis[(benzyloxy)methyl]uracil derivatives—Novel antivirals with activity against HIV-1 and influenza H1N1 virus

作者：Alexander N. Geisman^a ; Vladimir T. Valuev-Elliston^b ; Alexander A. Ozerov^a ; Anastasia L. Khandazhinskaya^b ; Alexander O. Chizhov^c ; Sergey N. Kochetkov^b ; Christophe Pannecouque^d ; Lieve Naesens^d ; Katherine L. Seley-Radtke^e ; ^{kseley@umbc.edu" class="auth_mail" title="E-mail the corresponding author} ; Mikhail S. Novikov^a

关键词：Uracil ; Non-nucleoside reverse transcriptase inhibitors ; NNRTIs ; HIV ; Influenza virus

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

9.Systematic evaluation of methyl ester bioisosteres in the context of developing alkenyldiarylmethanes (ADAMs) as non-nucleoside reverse transcriptase inhibitors (NNRTIs) for anti-HIV-1 chemotherapy

作者：Ayako Hoshi^a ; Takeshi Sakamoto^a ; ^{sakamoto@josai.ac.jp" class="auth_mail" title="E-mail the corresponding author} ; Jun Takayama^a ; Meiyan Xuan^a ; Mari Okazaki^a ; Tracy L. Hartman^b ; Robert W. Buckheit Jr.^b ; Christophe Pannecouque^c ; Mark Cushman^d ; ^{cushman@purdue.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：ADAM ; alkenyldiarylmethane ; NNRTI ; non-nucleoside reverse transcriptase inhibitor ; RT ; reverse transcriptase ; HIV-1 ; human immunodeficiency virus type 1 ; AIDS ; acquired immune deficiency syndrome ; ART ; antiretroviral therapy ; NRTI ; nucleoside reverse transcriptase inhibitor ; PI ; protease inhibitor ; INI ; integrase inhibitors ; FI ; fusion inhibitor ; CCR5I ; CC chemokine receptor inhibitor ; dNTPs ; deoxynucleoside triphosphate ; AZT ; azidothymidine (zidovudine) ; EDCI ; 1-(3-dimethylaminopropyl)-3-ethylc

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

10.Design, synthesis and anti-HIV activity of novel quinoxaline derivatives

作者：Saloni B. Patel^a ; Bhumika D. Patel^a ; Christophe Pannecouque^b ; Hardik G. Bhatt^a ; ^{hardikbhatt23@hotmail.com" class="auth_mail" title="E-mail the corresponding author}

关键词：AIDS ; HIV ; Pharmacophore modelling ; 3D-QSAR ; Quinoxaline

刊名：European Journal of Medicinal Chemistry

出版年：2016

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作者(114)

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2027年及以后(1)

2017年(1)

2016年(10)

2015年(2)

2013年(5)

2012年(9)

2011年(6)

2010年(9)

2009年(20)

2008年(10)

2007年(10)

2006年(4)

2004年(2)

2003年(2)

2002年(4)

2001年(3)

2000年(3)

2000年及以前(13)

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