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Wiley电子期刊(11)	NATURE电子期刊(2)	ACS电子期刊(57)
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在“Elsevier电子期刊”中，命中：683条，耗时：0.1699191 秒

在所有数据库中总计命中：945条

1.A new set of assays for the discovery of aminoacyl-tRNA synthetase inhibitors

作者：Adé ; laï ; de Saint-Lé ; ger^a ; Lluí ; s Ribas de Pouplana^a ; ^b ; ^c ; ^{lluis.ribas@irbbarcelona.org}

关键词：ARS ; aminoacyl-tRNA synthetases ; Cpd ; compound ; HTS ; high throughput screening ; IC50 ; half maximal inhibitory concentration ; Km ; Michaelis constant ; LRS ; leucyl-tRNA synthetase ; MIC ; minimum inhibitory concentration ; OM ; Omnia Molecular ; RLU ; relative light unit ; RRS ; arginyl-tRNA synthetase ; RT ; room temperature ; SRS ; seryl-tRNA synthetase ; SD ; standard deviation ; tRNA ; aminoacylate transfer RNA ; YRS ; tyrosyl-tRNA synthetase ; WRS ; tryptophanyl-tRNA synthetase ; Wt ; wild-type

刊名：Methods

出版年：2017

2.A data-driven weighting scheme for multivariate phenotypic endpoints recapitulates zebrafish developmental cascades

作者：Guozhu Zhang^a ; ^{gzhang6@ncsu.edu} ; Kyle R. Roell^a ; ^{krroell@ncsu.edu} ; Lisa Truong^c ; ^{lisa.truong@oregonstate.edu} ; Robert L. Tanguay^c ; ^{robert.tanguay@oregonstate.edu} ; David M. Reif^a ; ^b ; ^{dmreif@ncsu.edu}

关键词：AC50 ; half-maximal activity concentration ; AOP ; Adverse Outcome Pathway ; AggE ; Aggregate Entropy ; EZ ; embryonic zebrafish ; HTS ; high-throughput screening ; Hpf ; hours post fertilization ; LD50 ; 50% lethal dose ; MoA ; mechanisms of action ; POD ; point of departure ; ROC ; Receiver Operating Characteristic ; ToxRefDB ; Toxicity Reference Database ; wAggE ; weighted Aggregate Entropy ; TN ; true negative ; TP ; true positive ; FN ; false negative ; FP ; false negative ; MORT ; mortality ; YSE ; yolk sac edema ; AXIS ; bod

刊名：Toxicology and Applied Pharmacology

出版年：2017

3.Folic acid-decorated and PEGylated PLGA nanoparticles for improving the antitumour activity of 5-fluorouracil

作者：Mazen M. El-Hammadi^a ; ^b ; Á ; ngel V. Delgado^c ; Consolació ; n Melguizo^d ; ^e ; José ; C. Prados^d ; ^e ; José ; L. Arias^a ; ^d ; ^e ; ^{jlarias@ugr.es}

关键词：Cancer chemotherapy ; 5-Fluorouracil ; FOL-PEG-PLGA conjugate ; Haemocompatibility ; Ligand-receptor mediated drug delivery ; Nanoprecipitation.

刊名：International Journal of Pharmaceutics

出版年：2017

4.In vitro combinatory effects of the Alternaria mycotoxins alternariol and altertoxin II and potentially involved miRNAs

作者：Katharina Vejdovszky^a ; Matej Sack^b ; Katharina Jarolim^a ; Georg Aichinger^a ; Mark M. Somoza^b ; Doris Marko^a ; ^{doris.marko@univie.ac.at}

关键词：AOH ; alternariol ; ATX II ; altertoxin II miRNA microRNA ; ddPCR ; droplet digital polymerase chain reaction ; PBS ; phosphate buffered saline ; FBS ; fetal bovine serum ; DMSO ; dimethyl sulfoxide ; EC50 ; half maximal effective concentration ; SEM ; standard error of the mean ; SD ; standard error of the mean

刊名：Toxicology Letters

出版年：2017

5.Reassessing APOBEC3G Inhibition by HIV-1 Vif-Derived Peptides

作者：Christopher M. Richards¹ ; ² ; Ming Li¹ ; ² ; Angela L. Perkins³ ; ⁵ ; Anurag Rathore¹ ; ⁶ ; Daniel A. Harki³ ; Reuben S. Harris¹ ; ² ; ⁴ ; ^rsh@umn.edu

关键词：A3G ; APOBEC3G ; AID ; activation-induced deaminase ; CBF-β ; core-binding factor beta ; EMSA ; electrophoretic mobility shift assays ; G-to-A ; guanine-to-adenine ; HPLC ; high-performance liquid chromatography ; IC50 ; half maximal inhibitory concentration ; MS ; mass spectrometry ; PCR ; polymerase chain reaction ; ssDNA ; single-stranded DNA ; UDG ; uracil DNA glycosylase ; Vif ; viral infectivity factor

刊名：Journal of Molecular Biology

出版年：2017

6.Design, synthesis and analgesic/anti-inflammatory evaluation of novel diarylthiazole and diarylimidazole derivatives towards selective COX-1 inhibitors with better gastric profile

作者：Ahmed H. Abdelazeem^a ; ^b ; ^{ahmed.abdelazeem@pharm.bsu.edu.eg} ; ^{ahmed.pharm@yahoo.com} ; Mohammed T. El-Saadi^a ; Asmaa G. Safi El-Din^a ; Hany A. Omar^c ; ^d ; Samir M. El-Moghazy^e ; ^{samirelmoghazy@gmail.com}

关键词：Selective COX-1 ; Mofezolac ; Diarylthiazole ; Diarylimidazole ; Analgesic ; Anti-inflammatory ; Ulcerogenicity

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

7.Synthesis and bioactivities of novel 2-(thioether/sulfone)-5-pyrazolyl-1,3,4-oxadiazole derivatives

作者：Yu-Tao Zheng^a ; ¹ ; Teng-Teng Zhang^a ; ¹ ; Pei-Yi Wang^a ; Zhi-Bing Wu^a ; Lei Zhou^a ; Yi-Qiang Ye^a ; Xiang Zhou^a ; Ming He^a ; Song Yang^a ; ^b ; ^{jhzx.msm@gmail.com}

关键词：Pyrazole ; 13 ; 4-Oxadiazole ; Synthesis ; Antibacterial ; Antifungal

刊名：Chinese Chemical Letters

出版年：2017

8.Oestrogen reporter transgenic medaka for non-invasive evaluation of aromatase activity

作者：Petra Spirhanzlova^a ; ^c ; Mathilde Leleu^a ; Anthony Sé ; billot^a ; Gregory F. Lemkine^a ; ^{lemkine@watchfrog.fr" class="auth_mail" title="E-mail the corresponding author} ; Taisen Iguchi^b ; Barbara A. Demeneix^c ; Andrew J. Tindall^a

关键词：Tam ; Tamoxifen ; Fad ; Fadrozole ; Dex ; Dexamethasone ; T3 ; 3 ; 3&prime ; 5&prime ; -triiodo-l-thyronine ; EE2 ; 17α-ethinyl oestradiol ; E2 ; 17β-oestradiol ; EC50 ; Effective concentration 50 (half maximal effective concentration) ; T ; Testosterone ; SEM ; Standard error of the mean ; EDCs ; Endocrine disrupting chemicals ; ChgH ; Choriogenin H ; GFP ; Green fluorescent protein ; DMSO ; Dimethyl sulfoxide ; MS222 ; Ethyl 3-aminobenzoate methanesulfonate ; dph ; Day post hatch ; ER ; Oestrogen receptor ; SERM ; Selective oestro

刊名：Comparative Biochemistry and Physiology, Part C

出版年：2016

9.Vialinin A and thelephantin G, potent inhibitors of tumor necrosis factor-α production, inhibit sentrin/SUMO-specific protease 1 enzymatic activity

作者：Yasukiyo Yoshioka^a ; ^b ; Daisuke Namiki^a ; Mao Makiuchi^a ; Kouichi Sugaya^a ; Jun-ichi Onose^a ; Hitoshi Ashida^b ; ^c ; Naoki Abe^a ; ^{abe@nodai.ac.jp" class="auth_mail" title="E-mail the corresponding author}

关键词：cSENP1 ; catalytic human SUMO-specific protease ; DUB ; deubiquitinating enzyme ; IC50 ; half maximal inhibitory concentration ; rhSENP1 ; recombinant human SUMO-specific protease ; SENP ; SUMO-specific protease ; SUMO ; small ubiquitin-related protein modifier ; SUMO1-AMC ; SUMO1-7-amino-4-methylcoumarin ; TNFα ; tumor necrosis factor alpha ; USP5 ; ubiquitin-specific peptidase/isopeptidase ; NEM ; N-ethylamalemide

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

10.Structure activity relationship modelling of milk protein-derived peptides with dipeptidyl peptidase IV (DPP-IV) inhibitory activity

作者：Alice B. Nongonierma ; Richard J. FitzGerald ; ^{dick.fitzgerald@ul.ie" class="auth_mail" title="E-mail the corresponding author}

关键词：ACE ; angiotensin converting enzyme ; ANN ; artificial neural network ; BAP ; bioactive peptide ; BCAA ; branched chain amino acid ; β-Lg ; β-lactoglobulin ; BSA ; bovine serum albumin ; CN ; casein ; DPP-IV ; dipeptidyl peptidase IV ; GIP ; insulinotropic polypeptide ; GLP-1 ; glucagon-like peptide-1 ; HCl ; hydrochloric acid ; IC50 ; half maximal inhibitory concentration ; LF ; lactoferrin ; MLR ; multiple linear regression ; PCA ; principal component analysis ; PLSR ; partial least square regression ; pNA ; p-nitroanilide ; P

刊名：Peptides

出版年：2016

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