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Wiley电子期刊(3)	NATURE电子期刊(2)	ACS电子期刊(32)
SpringerLink电子期刊(37)	Elsevier电子期刊(97)

在“Elsevier电子期刊”中，命中：97条，耗时：0.1129461 秒

在所有数据库中总计命中：171条

1.Strategies for over-expression and purification of recombinant full length STAT5B in Escherichia coli

作者：Elvin D. de Araujo^a ; ^b ; Mulu Geletu^a ; ^b ; Patrick T. Gunning^a ; ^b ; ^{patrick.gunning@utoronto.ca" class="auth_mail" title="E-mail the corresponding author}

关键词：Recombinant Signal Transducer and Activator of Transcription 5B (STAT5B) expression ; Peptide fluorescence polarization ; Thermal shift assay ; Western blotting ; SYPRO Orange ; Osmolyte

刊名：Protein Expression and Purification

出版年：2017

2.Indole-3-carbinol (I3C) analogues are potent small molecule inhibitors of NEDD4-1 ubiquitin ligase activity that disrupt proliferation of human melanoma cells

作者：Jeanne G. Quirit^a ; ^{jgquirit@berkeley.edu} ; Sergey N. Lavrenov^b ; ^{satory@mail.ru} ; Kevin Poindexter^a ; ^{kpoindexter25@gmail.com} ; Janice Xu^a ; ^{jamicexu@scripps.edu} ; Christine Kyauk^a ; ^{ckyauk@berkeley.edu} ; Kathleen A. Durkin^c ; ^{durkin@berkeley.edu} ; Ida Aronchik^a ; ^{idaaronchik@gmail.com} ; Thomas Tomasiak^d ; ^{tomasiak@msg.ucsf.edu} ; Yaroslav A. Solomatin^b ; ^{hercules44@yandex.ru} ; Maria N. Preobrazhenskaya^b ; ^{satory@mail.ru} ; Gary L. Firestone^a ; ^{glfire@berkeley.edu}

关键词：Indole-3-carbinol analogues ; Ligand-target protein interactions ; NEDD4-1 ubiquitin ligase ; In silico computational modeling ; Anti-cancer compounds ; Melanoma cells

刊名：Biochemical Pharmacology

出版年：2017

3.Virtual screening and biophysical studies lead to HSP90 inhibitors

作者：Renjie Huang ; Daniel M. Ayine-Tora ; M. Nasri Muhammad Rosdi ; Yu Li ; Jó ; hannes Reynisson ; ^{j.reynisson@auckland.ac.nz} ; Ivanhoe K.H. Leung ; ^{i.leung@auckland.ac.nz}

关键词：17-AAG ; 17-allylamino-17-demethoxygeldanamycin ; 17-DMAG ; 17-(dimethylaminoethylamino)-17-demethoxygeldanamycin (17-DMAG) ; ADP ; adenosine diphosphate ; AMPPCP ; 5&prime ; -adenylylmethylenediphosphonate ; ASP ; Astex statistical potential ; ATP ; adenosine triphosphate ; CS ; ChemScore ; GS ; GoldScore ; HB ; hydrogen bonding ; HSP90 ; heat shock protein 90 ; HSQC ; heteronuclear single quantum correlation ; KD ; binding affinity ; ND ; N-domain ; NMR ; nuclear magnetic resonance ; NOE ; nuclear Overhauser effect ; Tm ; pro

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

4.Structure-guided discovery of thiazolidine-2,4-dione derivatives as a novel class of Leishmania major pteridine reductase 1 inhibitors

作者：Franco Henrique A. Leite^a ; Priscila Brandã ; o Gomes da Silva Santiago^b ; Thamires Quadros Froes^d ; Joã ; o da Silva Filho^b ; Suellen Gonç ; alves da Silva^d ; Rafael M. Ximenes^b ; Antô ; nio Rodolfo de Faria^c ; Dalci José ; Brondani^c ; Julianna F.C. de Albuquerque^b ; Marcelo Santos Castilho^a ; ^d ; ^{castilho@ufba.br" class="auth_mail" title="E-mail the corresponding author}

关键词：Leishmania ; Thiazolidine-2 ; 4-dione derivatives ; Pteridine reductase 1 ; Thermal shift assay ; Kinetic assay ; Molecular modeling

刊名：European Journal of Medicinal Chemistry

出版年：2016

5.Increasing the spectral shifts in LSPR biosensing using DNA-functionalized gold nanorods in a competitive assay format for the detection of interferon-γ

作者：Ding-Zheng Lin^a ; Po-Chun Chuang^b ; Pei-Chen Liao^c ; Jung-Po Chen^d ; Yih-Fan Chen^b ; ^e ; ^{chenyf@ym.edu.tw" class="auth_mail" title="E-mail the corresponding author}

关键词：Localized surface plasmon resonance ; Gold nanorod ; Aptamer ; Interferon gamma ; Label free

刊名：Biosensors and Bioelectronics

出版年：2016

6.Intrinsic thermodynamics of inhibitor binding to human carbonic anhydrase IX

作者：Vaida Linkuvienė ; Jurgita Matulienė ; Vaida Juozapaitienė ; Vilma Michailovienė ; Jelena Jachno ; Daumantas Matulis ; ^{daumantas.matulis@bti.vu.lt" class="auth_mail" title="E-mail the corresponding author} ; ^{matulis@ibt.lt" class="auth_mail" title="E-mail the corresponding author}

关键词：Intrinsic thermodynamics of protein-ligand binding ; Carbonic anhydrase ; Benzenesulfonamide inhibitors ; Fluorescent thermal shift assay ; Isothermal titration calorimetry ; Drug design

刊名：Biochimica et Biophysica Acta (BBA) - General Subjects

出版年：2016

7.Novel small molecule binders of human N-glycanase 1, a key player in the endoplasmic reticulum associated degradation pathway

作者：Bharath Srinivasan ^{bharath.srinivasan@biology.gatech.edu" class="auth_mail" title="E-mail the corresponding author} ; Hongyi Zhou ; Sreyoshi Mitra ; Jeffrey Skolnick ; ^{skolnick@gatech.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：NGLY1 ; N-glycanase ; ER ; endoplasmic reticulum ; ERAD ; endoplasmic reticulum associated degradation ; SDS&ndash ; PAGE ; sodium dodecyl sulfate polyacrylamide gel electrophoresis ; TSA ; thermal shift assay ; DSF ; differential scanning fluorimetry

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

8.Thermodynamic properties of leukotriene A₄ hydrolase inhibitors

关键词：LTA4H ; leukotriene A4 hydrolase ; LTA4 ; leukotriene A4 ; LTB4 ; leukotriene B4 ; kDa ; kilo Dalton ; PGP ; prolin&ndash ; glycin&ndash ; prolin ; TSA ; thermal shift assay ; TM ; melting point ; ITC ; isothermal titration calorimetry ; DSF ; different scanning fluorimetry ; Ki ; inhibitory constant ; Kd ; dissoziation constant

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

9.Identification of B. anthracis N⁵-carboxyaminoimidazole ribonucleotide mutase (PurE) active site binding compounds via fragment library screening

作者：Hao Lei^a ; Christopher Jones^a ; Tian Zhu^a ; Kavankumar Patel^a ; Nina M. Wolf^b ; Leslie W.-M. Fung^b ; Hyun Lee^a ; ^{danielhl@uic.edu" class="auth_mail" title="E-mail the corresponding author} ; Michael E. Johnson^a ; ^{mjohnson@uic.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：PurE ; N5-carboxyaminoimidazole ribonucleotide mutase ; FBDD ; fragment-based drug design ; NMR ; nuclear magnetic resonance ; STD-NMR ; saturation transfer difference nuclear magnetic resonance (NMR) ; WaterLOGSY NMR ; water ligand observed via gradient spectroscopy NMR ; SPR ; surface plasmon resonance ; TSA ; thermal shift assay ; N5-CAIR ; N5-carboxyaminoimidazole ribonucleotide ; CAIR ; 4-carboxyaminoimidazole ribonucleotide ; AIR ; aminoimidazole ribonucleotide

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

10.Andrographolide reversed 5-FU resistance in human colorectal cancer by elevating BAX expression

作者：Weicheng Wang^a ; ¹ ; Wenjie Guo^b ; ¹ ; Lele Li^a ; ¹ ; Zan Fu^a ; Wen Liu^b ; Jian Gao^b ; Yongqian Shu^a ; Qiang Xu^b ; ^{molpharm@163.com" class="auth_mail" title="E-mail the corresponding author} ; Yang Sun^b ; ^{yangsun@nju.edu.cn" class="auth_mail" title="E-mail the corresponding author} ; Yanhong Gu^a ; ^{guyhphd@163.com" class="auth_mail" title="E-mail the corresponding author}

关键词：Andrographolide ; BAX ; 5-FU-resistant ; Human colorectal cancer

刊名：Biochemical Pharmacology

出版年：2016

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