作者：M.J. Gó ; mara^a ; ^{mariajose.gomara@iqac.csic.es" class="auth_mail" title="E-mail the corresponding author} ; V. Sá ; nchez-Merino^b ; A. Paú ; s^a ; A. Merino-Mansilla^b ; J.M. Gatell^b ; ^c ; E. Yuste^b ; I. Haro^a ; ^{isabel.haro@iqac.csic.es" class="auth_mail" title="E-mail the corresponding author}

关键词：Acm ; acetamidomethyl ; ACN ; acetonitrile ; Dbz ; diaminobenzoyl ; DHB ; 2 ; 5-dihydroxybenzoic acid ; DIPEA ; diisopropylethylamine ; FP ; fusion peptide ; GBV-C ; GB virus C ; HAART ; highly active antiretroviral therapy ; HATU ; 2-(1H-7-azabenzotriazole-1-yl)-113 ; 3-tetramethyluronium hexafluorophosphate methanaminium ; HB ; helix bundle ; HT ; head-to-tail ; LUV ; large unilamelar vesicles ; mAb ; monoclonal antibody ; MPAA ; 4-mercaptophenylacetic acid ; MPER ; membrane proximal external region ; NBD ; 6-(7-nitrobenzofur

刊名：Biochimica et Biophysica Acta (BBA) - General Subjects

出版年：2016

作者：Nicholas S. Kirk^a ; Anna Bezos^b ; Anthony C. Willis^c ; Pichit Sudta^d ; ^e ; Sunit Suksamrarn^e ; Christopher R. Parish^b ; Marie Ranson^f ; Michael J. Kelso^a ; ^{mkelso@uow.edu.au" class="auth_mail" title="E-mail the corresponding author}

关键词：HBTU ; 2-(1H-benzotriazol-1-yl)-113 ; 3-tetramethyluronium hexafluorophosphate ; CSF-1R ; colony-stimulating factor-1 receptor ; DIPEA ; N ; N-diisopropylethylamine ; FLT-3 ; Fms-like tyrosine kinase 3 ; FOV ; field of view ; HUVEC ; human umbilical vein endothelial cell ; PDGFR ; platelet-derived growth factor receptor ; RTK ; receptor tyrosine kinase ; THF ; tetrahydrofuran ; VEGFR ; vascular endothelial growth factor receptor

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

作者：Takuya Arai^a ; ^b ; Akiko Ohno^c ; Kazunori Mori^b ; Hiroshi Kuwata^b ; Mirei Mizuno^b ; Kohei Imai^b ; Shuntaro Hara^b ; Motoko Shibanuma^b ; Masaaki Kurihara^c ; Naoki Miyata^a ; Hidehiko Nakagawa^a ; Kiyoshi Fukuhara^b ; ^{fukuhara@pharm.showa-u.ac.jp" class="auth_mail" title="E-mail the corresponding author}

关键词：Aβ ; amyloid-β ; AD ; Alzheimer&rsquo ; s disease ; CA ; caffeic acid ; DCFH-DA ; 2&prime ; 7&prime ; -dichlorodihydrofluorescein diacetate ; DHCA ; dihydrocaffeic acid ; DIPEA ; N ; N-diisopropylethylamine ; DMF ; N ; N-dimethylformamide ; DMSO ; dimethyl sulfoxide ; Gly ; glycine ; HBTU ; O-(benzotriazol-1-yl)- NN ; N&prime ; N&prime ; -tetramethyluronium hexafluorophosphate ; HFIP ; 11133 ; 3-hexafluoro-2-propanol ; HOBt ; 1-hydroxybenzotriazole ; HRMS ; high resolution mass spectrometry ; PI ; propidium iodide ; ROS ; reactive oxy

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

作者：Lauren E. Ragle^a ; Dilip J. Palanisamy^a ; Margaux J. Joe^a ; Rachel S. Stein^a ; Derek D. Norman^b ; Gabor Tigyi^b ; Daniel L. Baker^a ; Abby L. Parrill^a ;

关键词：ATX/NPP2 ; autotaxin ; DIPEA ; N ; N-diisopropylethylamine ; DMF ; N ; N-dimethylformamide ; DMSO ; dimethylsulfoxide ; GPCR ; G-protein coupled receptor ; GRI ; Genomic Research Institute ; HBTU ; O-(benzotriazol-1-yl)-NN ; N&prime ; N&prime ; -tetramethyluronium hexafluorophosphate ; LPC ; lysophosphatidylcholine ; LPA ; lysophosphatidic acid ; LysoPLD ; lysophospholipase-D ; MOE ; Molecular Operating Environment ; NPP ; nucleotide pyrophosphatase phosphodiesterase ; pNP-TMP ; p-nitrophenyl thymidine-5&prime ; -monophosphate ; p

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

作者：Dražen Pavlović ; ^{dpavlovic@hotmail.fr" class="auth_mail" title="E-mail the corresponding author} ; Stjepan Mutak

关键词：MLSB ; macrolide&ndash ; lincosamide&ndash ; streptogramin B antibiotics ; HBTU ; O-(benzotriazol-1-yl)-NN ; N&prime ; N&prime ; -tetramethyluronium hexafluorophosphate ; DIPEA ; diisopropylethylamine ; SAR ; structure&ndash ; activity relationships

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

作者：Takaharu Hirayama ; ^{takaharu.hirayama@takeda.com" class="auth_mail" title="E-mail the corresponding author} ; Masanori Okaniwa ; ^{masanori.okaniwa@takeda.com" class="auth_mail" title="E-mail the corresponding author} ; Hiroshi Banno ; Hiroyuki Kakei ; Akihiro Ohashi ; Momoko Ohori ; Tadahiro Nambu ; Kenichi Iwai ; Tomohiro Kawamoto ; Akihiro Yokota ; Maki Miyamoto ; Tomoyasu Ishikawa

关键词：DIPEA ; N ; N-diisopropylethylamine ; HATU ; hexafluorophosphate O-(7-azabenzotriazol-1-yl)-NN ; N&prime ; N&prime ; -tetramethyluronium ; PD ; pharmacodynamic

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2016

作者：Takuya Arai^a ; ^b ; Akiko Ohno^c ; Mori Kazunori^b ; Taeko Kakizawa^c ; Hiroshi Kuwata^b ; Toshihiko Ozawa^d ; Motoko Shibanuma^b ; Shuntaro Hara^b ; Seiichi Ishida^e ; Masaaki Kurihara^c ; Naoki Miyata^a ; Hidehiko Nakagawa^a ; Kiyoshi Fukuhara^b ; ^{fukuhara@pharm.showa-u.ac.jp" class="auth_mail" title="E-mail the corresponding author}

关键词：AA ; amino acid ; Aβ ; amyloid-β ; AD ; Alzheimer&rsquo ; s disease ; DCFH-DA ; 2&prime ; 7&prime ; -dichlorodihydrofluorescein diacetate ; DIPEA ; N ; N-diisopropylethylamine ; DMF ; N ; N-dimethylformamide ; DMSO ; dimethyl sulfoxide ; HBTU ; O-(benzotriazol-1-yl)-NN ; N&prime ; N&prime ; -tetramethyluronium hexafluorophosphate ; HFIP ; 11133 ; 3-hexafluoro-2-propanol ; HOBt ; 1-hydroxybenzotriazole ; HRMS ; high resolution mass spectrometry ; PI ; propidium iodide ; ROS ; reactive oxygen species ; RP-HPLC ; reverse phase high per

刊名：Bioorganic & Medicinal Chemistry

出版年：2016

作者：M.F.M. Marcondes ; F.M. Alves ; D.M. Assis¹ ; I.Y. Hirata ; L. Juliano ; V. Oliveira ; ^{vitor.oliveira@unifesp.br" class="auth_mail" title="E-mail the corresponding author} ; M.A. Juliano ; ^{ma.juliano@unifesp.br" class="auth_mail" title="E-mail the corresponding author}

关键词：Abz ; ortho-aminobenzoic acid ; EDDnp ; N-(2 ; 4-dinitrophenyl)-ethylenediamine ; FRET ; fluorescence resonance energy transfer ; hMIP ; human mitochondrial intermediate peptidase ; HOBt ; hydroxybenzotriazole ; TBTU ; O-(benzotriazol-1-yl)-NN ; N&prime ; N&prime ; -tetramethyluronium tetrafluoroborate ; NMM ; N-methylmorpholine ; DMF ; dimethylformamide ; DIPEA ; N ; N-diisopropylethylamine ; DCM ; dichloromethane

刊名：FEBS Open Bio

出版年：2015

作者：Sofia Zanin^a ; Michele Sandre^b ; Giorgio Cozza^a ; Daniele Ottaviani^a ; Oriano Marin^a ; ^b ; ^{oriano.marin@unipd.it" class="auth_mail" title="E-mail the corresponding author} ; Lorenzo A. Pinna^a ; ^c ; Maria Ruzzene^a ; ^{maria.ruzzene@unipd.it" class="auth_mail" title="E-mail the corresponding author}

关键词：Akt ; protein kinase Akt (PKB) ; B23 ; nucleophosmin ; BSA ; bovine serum albumin ; CaM ; calmodulin ; CK2-MCP ; CK2 modulatory chimeric peptide ; CK2 ; protein kinase CK2 ; (casein kinase 2) ; CM5 ; carboxymethylated dextran 5 ; CML ; chronic myeloid leukemia ; DC50 ; concentration inducing 50% cell death ; DMEM ; Dulbecco's Modified Eagle's Medium ; DTT ; dithiothreitol ; eiF2β ; elongation initiation factor 2β ; FBS ; fetal bovine serum ; HATU ; O-(7-azabenzotriazole-1-yl)-NNN ; N&prime ; -tetramethyluronium hexafluoropho

刊名：Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics

出版年：2015

作者：A. Gauna^a ; ^{adrygauna@gmail.com" class="auth_mail" title="E-mail the corresponding author} ; S. Losada^a ; ^{salosada@yahoo.com" class="auth_mail" title="E-mail the corresponding author} ; M. Lorenzo^a ; ^{angelita.lorenzo@gmail.com" class="auth_mail" title="E-mail the corresponding author} ; H. Bermú ; dez^a ; ^{henrybermudez2001@yahoo.com" class="auth_mail" title="E-mail the corresponding author} ; M. Toledo^b ; ^{marilyan@gmail.com" class="auth_mail" title="E-mail the corresponding author} ; H. Pé ; rez^c ; ^{hperez113@hotmail.com" class="auth_mail" title="E-mail the corresponding author} ; E. Chacó ; n^c ; ^{elsach7@hotmail.com" class="auth_mail" title="E-mail the corresponding author} ; O. Noya^a ; ^d ; ^{noyaoo@yahoo.com" class="auth_mail" title="E-mail the corresponding author}

关键词：NMP ; N-Methyl-2-pyrrolidone ; HOBt ; hydroxybenzotriazole ; DIC ; N ; N&prime ; -Diisopropylcarbodiimide ; TFA ; trifluoroacetic acid ; DCM ; dichloromethane ; TIPS ; triisopropylsilane ; TBTU ; 2-(1H-Benzotriazol-1-yl)-113 ; 3-tetramethyluroniumtetrafluoroborate ; DMSO ; dimethyl sulfoxide ; PBS ; phosphate buffered saline ; IMT ; Instituto de Medicina Tropical

刊名：Journal of Immunological Methods

出版年：2015