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Wiley电子期刊(10)	NATURE电子期刊(15)	ACS电子期刊(79)
SpringerLink电子期刊(233)	Elsevier电子期刊(2087)

在“Elsevier电子期刊”中，命中：2,087条，耗时：0.0399806 秒

在所有数据库中总计命中：2,424条

1.Synthesis of novel steroidal agonists, partial agonists, and antagonists for the glucocorticoid receptor

作者：Zhuang Jin^a ; Hua Lin^a ; Sathish Srinivasan^b ; Jerome C. Nwachukwu^b ; Nelson Bruno^b ; Patrick R. Griffin^a ; Kendall W. Nettles^b ; ; Theodore M. Kamenecka^a ; ^{kameneck@scripps.edu}

关键词：AF-1 ; activation function-1 ; AF-2 ; activation function-2 ; AP-1 ; activator protein 1 ; dppp ; 1 ; 3-bis(diphenylphosphino)propane ; DEX ; dexamethasone ; DIEA ; N ; N-diisopropylethylamine ; FKBP5 ; FK506-binding protein 5 ; GR ; glucocorticoid receptor ; GRE ; glucocorticoid-response element ; HATU ; 1-[bis(dimethylamino)methylene]-1H-12 ; 3-triazolo[4 ; 5-b]pyridinium 3-oxid hexafluorophosphate ; IL-6 ; Interleukin-6 ; LBD ; ligand-binding domain ; LPS ; lipopolysaccharide ; MMTV ; mouse mammary tumor virus ; NF-κB ; nuclear

刊名：Bioorganic & Medicinal Chemistry Letters

出版年：2017

2.Naturally-occurring TGR5 agonists modulating glucagon-like peptide-1 biosynthesis and secretion

作者：Laila Jafri^a ; ^d ; ² ; ^{lailashah9@gmail.com" class="auth_mail" title="E-mail the corresponding author} ; Samreen Saleem^b ; ^d ; ^{samreen.qau@gmail.com" class="auth_mail" title="E-mail the corresponding author} ; Danielle Calderwood^c ; ^{dcalderwood01@qub.ac.uk" class="auth_mail" title="E-mail the corresponding author} ; Anna Gillespie^c ; ^{agillespie14@qub.ac.uk" class="auth_mail" title="E-mail the corresponding author} ; Bushra Mirza^d ; ¹ ; ^{bushramirza@qau.edu.pk" class="auth_mail" title="E-mail the corresponding author} ; Brian D. Green^c ; ¹ ; ^{b.green@qub.ac.uk" class="auth_mail" title="E-mail the corresponding author}

关键词：GLP-1 ; GIP ; Incretin ; Secretagogue ; TGR5

刊名：Peptides

出版年：2016

3.The triterpene echinocystic acid and its 3-O-glucoside derivative are revealed as potent and selective glucocorticoid receptor agonists

作者：Demetra Georgatza^a ; ¹ ; Vyron A. Gorgogietas^a ; ¹ ; Paraskevi Kylindri^a ; Maria Ch. Charalambous^a ; Kalliope K. Papadopoulou^a ; Joseph M. Hayes^b ; Anna-Maria G. Psarra^a ; ^{ampsarra@bio.uth.gr" class="auth_mail" title="E-mail the corresponding author} ; ^{ampsarra@gmail.com" class="auth_mail" title="E-mail the corresponding author}

关键词：GCs ; glucocorticoids ; GR ; glucocorticoid receptor ; SEGRA ; selective glucocorticoid receptor agonist ; EA ; echinocystic acid ; EA-3G ; echinocystic acid 3-O-glucoside ; PEPCK ; phosphoenolpyruvate carboxykinase ; NF-κB ; nuclear factor kappa beta ; TNF α ; tumour necrosis factor alpha ; CMX ; mito tracker red CMXRos ; DEX ; dexamethasone ; DAC ; deacylcortivazol ; GREs ; glucocorticoid responsive elements ; LBD ; ligand binding domain ; HPA ; hypothalamic&ndash ; pituitary&ndash ; adrenal ; RLU ; relative luciferase units

刊名：International Journal of Biochemistry and Cell Biology

出版年：2016

4.GnRH-agonist implantation of prepubertal male cats affects their reproductive performance and testicular LH receptor and FSH receptor expression

作者：N.S. Mehl^a ; M. Khalid^b ; S. Srisuwatanasagul^c ; T. Swangchan-uthai^a ; S. Sirivaidyapong^a ; ^{sudson.s@chula.ac.th" class="auth_mail" title="E-mail the corresponding author}

关键词：GnRH-agonist ; Prepubertal cat ; LHR ; FSHR ; Reproductive behavior

刊名：Theriogenology

出版年：2016

5.Berberine attenuates high glucose-induced fibrosis by activating the G protein-coupled bile acid receptor TGR5 and repressing the S1P2/MAPK signaling pathway in glomerular mesangial cells

作者：Zhiying Yang^a ; ^c ; ¹ ; Jie Li^b ; ¹ ; Fengxiao Xiong^a ; Junying Huang^a ; Cheng Chen^a ; Peiqing Liu^a ; ^c ; Heqing Huang^a ; ^b ; ^c ; ^{huangheq@mail.sysu.edu.cn" class="auth_mail" title="E-mail the corresponding author}

关键词：AP-1 ; active protein-1 ; BBR ; berberine ; DN ; diabetic nephropathy ; ERK ; extracellular signal-regulated kinase ; FN ; fibronectin ; GMCs ; glomerular mesangial cells ; ICAM-1 ; intercellular adhesion molecule-1 ; JNK ; c-Jun-NH2-terminal kinase ; MAPK ; mitogen-activated protein kinase ; S1P ; sphingosine 1-phosphate ; S1P2 ; sphingosine 1-phosphate receptor 2 ; Sphk1 ; sphingosine kinase ; TGF-β1 ; transforming growth factor-beta 1 ; TGR5 ; takeda G -protein-coupled receptor 5

刊名：Experimental Cell Research

出版年：2016

6.Effect of housing density on growth, agonistic behaviour, and activity in hatchling saltwater crocodiles (Crocodylus porosus)

作者：Matthew L. Brien^a ; ^b ; ^{matthew_brien@hotmail.com" class="auth_mail" title="E-mail the corresponding author} ; Grahame J. Webb^a ; ^b ; Keith A. McGuinness^a ; Keith A. Christian^a

关键词：Agonistic behaviour ; Hatchlings ; Density ; Activity ; Growth

刊名：Applied Animal Behaviour Science

出版年：2016

7.The neuroprotective effects of orthosteric agonists of group II and III mGluRs in primary neuronal cell cultures are dependent on developmental stage

作者：D. Jantas^a ; ^{jantas@if-pan.krakow.pl" class="auth_mail" title="E-mail the corresponding author} ; A. Gręda^a ; S. Gołda^b ; M. Korostyński^b ; W. Lasoń^a

关键词：ACPT-I ; LY354740 ; VU0361737 ; AMN082 ; Staurosporine ; Doxorubicin ; Glutamate ; Primary neuronal cell cultures

刊名：Neuropharmacology

出版年：2016

8.LXRα represses LPS-induced inflammatory responses by competing with IRF3 for GRIP1 in Kupffer cells

作者：Chun-mu Miao^a ; Kun He^a ; Pei-zhi Li^a ; Zuo-jin Liu^a ; Xi-wen Zhu^a ; Zhi-bing Ou^a ; Xiong-zhong Ruan^b ; Jian-ping Gong^a ; Chang-an Liu^a ; ^{liuchangan120@163.com" class="auth_mail" title="E-mail the corresponding author}

关键词：Liver X receptor ; Kupffer cell ; Interferon regulatory factor 3 ; Glucocorticoid receptor-interacting protein 1 ; Nuclear factor-kappa B

刊名：International Immunopharmacology

出版年：2016

9.Progestin-mediated activation of MAPK and AKT in nuclear progesterone receptor negative breast epithelial cells: The role of membrane progesterone receptors

作者：Monica Salazar^a ; ^{smony@nmsu.edu" class="auth_mail" title="E-mail the corresponding author} ; Alejandra Lerma-Ortiz^a ; ^{alelerma@nmsu.edu" class="auth_mail" title="E-mail the corresponding author} ; Grace M. Hooks^b ; ^{ghooks@nmsu.edu" class="auth_mail" title="E-mail the corresponding author} ; Amanda K. Ashley^b ; ^{ashleyak@nmsu.edu" class="auth_mail" title="E-mail the corresponding author} ; Ryan L. Ashley^a ; ^{ryashley@nmsu.edu" class="auth_mail" title="E-mail the corresponding author}

关键词：P4 ; progesterone ; MPR ; membrane progesterone receptor ; MPR-Ag ; membrane progesterone receptor agonist ; PR ; nuclear progesterone receptor ; MPA ; medroxyprogesterone acetate ; 5αP ; 5α-dihydroprogesterone ; 3αHP ; 3α-dihydroprogesterone ; PGRMC1 ; progesterone receptor membrane component-1 ; CHT ; combined hormone therapy (estrogen ; + ; progestin) ; EHT ; unopposed estrogen hormone therapy

刊名：Gene

出版年：2016

10.Parcours de soins du patient adulte souffrant de syndrome de grêle court avec insuffisance intestinale

作者：Francisca Joly^a ; ^b ; ^c ; ^{francisca.joly@bjn.aphp.fr} ; Vanessa Boehm^a ; ^b ; Julie Bataille^a ; ^b ; ^d ; Lore Billiauws^a ; ^b ; Olivier Corcos^b ; ^e ; la Commission nutrition et parcours de soins de la SFNEP¹

关键词：É ; quilibre hydroé ; lectrolytique ; Nutrition parenté ; rale ; Nutrition enté ; rale ; Ré ; instillation du chyme digestif ; Facteurs trophiques intestinaux

刊名：Nutrition Clinique et Métabolisme

出版年：2016

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