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中国地质文献-英文(2)	SpringerLink电子期刊(13852)	NATURE电子期刊(92)	Elsevier电子期刊(42741)
Wiley电子期刊(416)	ProQuest学位论文(25)	GSW全文库(59)	ACS电子期刊(4019)

在“Elsevier电子期刊”中，命中：42,741条，耗时：0.2179248 秒

在所有数据库中总计命中：61,206条

1.Ro 90-7501 inhibits PP5 through a novel, TPR-dependent mechanism

作者：Tae-Joon Hong^a ; Kwanghyun Park^a ; Eun-Wook Choi^b ; Ji-Sook Hahn^a ; ^{hahnjs@snu.ac.kr}

关键词：Protein phosphatase 5 (PP5) ; Ro 90-7501 ; Inhibitor screening ; TPR-dependent inhibition

刊名：Biochemical and Biophysical Research Communications

出版年：2017

2.Treatment of estrogen-dependent diseases: Design, synthesis and profiling of a selective 17β-HSD1 inhibitor with sub-nanomolar IC₅₀ for a proof-of-principle study

作者：Ahmed S. Abdelsamie^a ; ^b ; Chris J. van Koppen^c ; Emmanuel Bey^c ; Mohamed Salah^a ; Carsten Bö ; rger^d ; Lorenz Siebenbü ; rger^d ; Matthias W. Laschke^e ; Michael D. Menger^e ; Martin Frotscher^a ; ^{m.frotscher@mx.uni-saarland.de}

关键词：17β-Hydroxysteroid dehydrogenase type 1 ; Enzyme inhibitor ; Steroidogenic enzymes ; Estrogen-dependent disease ; Intracrinology

刊名：European Journal of Medicinal Chemistry

出版年：2017

3.Anti-angiogenic potential of trypsin inhibitor purified from Cucumis melo seeds: Homology modeling and molecular docking perspective

作者：Hassan Rasouli^a ; Sharham Parvaneh^a ; Azadeh Mahnam^a ; Mohsen Rastegari-Pouyani^b ; Zohreh Hoseinkhani^a ; Kamran Mansouri^a ; ^{kmansouri@kums.ac.ir} ; ^{kamranmansouri@gmail.com}

关键词：BSA ; bovine serum albumin ; DMEM ; Dulbecco&rsquo ; s modified eagle&rsquo ; s medium ; BBI ; Bowman-Birk inhibitor ; ELISA ; enzyme-linked immunosorbent assay ; FBS ; fetal bovine serum ; HUVEC ; human umbilical vein endothelial cells ; LDH ; lactate dehydrogenase ; MTT ; 3-(4 ; 5-dimethylthiazol-2yl)-2 ; 5-diphenyl-2H-tetrazolium bromide ; PBS ; phosphate buffered saline ; PBST ; PBS containing tween 20 ; PDB ; protein data bank ; SDS-PAGE ; sodium dodecyl sulfate polyacrylamide gel electrophoresis ; TICMS ; trypsin inhibito

刊名：International Journal of Biological Macromolecules

出版年：2017

4.Synthesis of novel β-propanamides to inhibit cholesteryl ester transfer protein (CETP)

作者：Hong-Lei Xie ; Chun-Chi Liu ; Yi-Qun Li ; Chang-Lin Bai ; Chen-Zhou Hao ; Jing Guo ; Chang-Qun Luo ; Dong-Mei Zhao ; ^{medchemzhao@163.com} ; Mao-Sheng Cheng

关键词：CETP inhibitor ; Cardiovascular disease ; High-density lipoprotein ; Low-density lipoprotein ; In vitro

刊名：Chinese Chemical Letters

出版年：2017

5.MiR-509-5p suppresses the proliferation, migration, and invasion of non-small cell lung cancer by targeting YWHAG

作者：Peng Wang ; Yu Deng ; ^{Leojokea@aliyun.com} ; XiangNing Fu ; ^{fuxn2006@aliyun.com}

关键词：Non-small lung cancer (NSCLC) ; MiR-509-5p ; YWHAG ; Akt

刊名：Biochemical and Biophysical Research Communications

出版年：2017

6.Long non-coding RNA NEAT1 facilitates pancreatic cancer progression through negative modulation of miR-506-3p

作者：Bo Huang^a ; ¹ ; Chuan Liu^b ; ¹ ; Qiong Wu^a ; Jing Zhang^a ; Qinghua Min^a ; Tianle Sheng^b ; Xiaozhong Wang^a ; Yeqing Zou^b ; ^{zouyeqing3366@163.com}

关键词：Pancreatic cancer ; Cell proliferation ; LncRNA NEAT1 ; miR-506-3p

刊名：Biochemical and Biophysical Research Communications

出版年：2017

7.Evaluation of additive formulations to inhibit precipitation of positive electrolyte in vanadium battery

作者：Faizur Rahman^a ; ^{rahman.faiz@gmail.com} ; M. Skyllas-Kazacos^b ; ^{M.Kazacos@unsw.edu.au}

关键词：Vanadium battery ; Positive vanadium electrolyte ; Scale inhibitor ; Additive ; V(V) precipitation

刊名：Journal of Power Sources

出版年：2017

8.Inhibition kinetics and molecular simulation of p-substituted cinnamic acid derivatives on tyrosinase

作者：Yi Cui^a ; Yong-Hua Hu^a ; Feng Yu^a ; Jing Zheng^a ; Lin-Shan Chen^a ; Qing-Xi Chen^a ; ^b ; Qin Wang^a ; ^{qwang@xmu.edu.cn}

关键词：4-CCA ; 4-chlorocinnamic acid ; 4-ECA ; 4-ethoxycinnamic acid ; 4-NCA ; 4-nitrocinnamic acid ; DMSO ; dimethyl-sulfoxide ; L-Tyr ; L-tyrosine ; L-DOPA ; L-3 ; 4-Dihydroxyphenylalanine ; Km ; Michaelis-Menten constant ; KI ; equilibrium constant of the inhibitor combining with the free enzyme ; IC50 ; inhibitor concentration leading to a 50% loss of activity

刊名：International Journal of Biological Macromolecules

出版年：2017

9.Phase 2 Study of Erlotinib in Combination With Linsitinib (OSI-906) or Placebo in Chemotherapy-Naive Patients With Non-Small-Cell Lung Cancer and Activating Epidermal Growth Factor Receptor Mutations

作者：Natasha B. Leighl¹ ; Naiyer A. Rizvi² ; Lopes Gilberto de Lima Jr.³ ; ⁴ ; Wichit Arpornwirat⁵ ; Charles M. Rudin⁶ ; Alberto A. Chiappori⁷ ; Myung-Ju Ahn⁸ ; Laura Q.M. Chow⁹ ; Lyudmila Bazhenova¹⁰ ; Arunee Dechaphunkul¹¹ ; Patrapim Sunpaweravong¹² ; Keith Eaton¹³ ; ¹⁴ ; Jihong Chen¹⁵ ; Sonja Medley¹⁵ ; Srinivasu Poondru¹⁵ ; Margaret Singh¹⁵ ; Joyce Steinberg¹⁵ ; Rosalyn A. Juergens¹⁶ ; ^{juergensr@hhsc.ca} ; Shirish M. Gadgeel¹⁷ ; ¹⁸

关键词：Combination ; Epidermal growth factor receptor inhibitor ; First-line therapy ; Insulin-like growth factor-1 inhibitor ; Tyrosine kinase inhibitor

刊名：Clinical Lung Cancer

出版年：2017

10.Regulation of merlin by protein phosphatase 1-TIMAP and EBP50 in endothelial cells

作者：Anita Boratkó ; ¹ ; Margit Pé ; ter¹ ; Csilla Csortos ; ^{csortos@med.unideb.hu}

关键词：BPAEC ; Bovine Pulmonary Artery Endothelial Cells ; ERM ; ezrin ; radixin ; moesin ; FERM ; band 4.1 ; ezrin ; radixin ; moesin ; GST ; glutathione S-transferase ; ILK ; integrin-linked kinase ; IP ; immunoprecipitation ; MYPT ; myosin phosphatase target subunit ; NF2 ; neurofibromatosis type 2 ; NHERF ; Na+/H+ exchanger regulatory factor ; PAK ; p21-activated kinase ; PKA ; cAMP-dependent protein kinase ; PKC ; protein kinase C ; PP ; protein phosphatase ; PP1c ; catalytic subunit of PP1 ; PP1c-MYPT1 ; myosin phosphatase ; TIMAP

刊名：The International Journal of Biochemistry & Cell Biology

出版年：2017

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